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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T4390 | ML221 | Apelin receptor , Arrestin | |
ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in the β-arrestin assay, and EC80 of 10 nM in both assays. |