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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T63014 | Ivabradine | ||
Ivabradine is a potent, orally active HCN (hyperpolarization-activated cyclic nucleotide-gated) channel blocker that inhibits pacemaker current (If). ivabradine decreases heart rate in a dose-dependent manner and does no... | |||
T2535 | Ivabradine hydrochloride | S 16257-2,Ivabradine HCl | Adrenergic Receptor |
Ivabradine hydrochloride (S 16257-2) is a new If inhibitor (IC50: 2.9 μM). Ivabradine Hydrochloride is the hydrochloride salt form of ivabradine, an orally bioavailable, hyperpolarization-activated, cyclic nucleotide-gat... | |||
T11692 | Ivabradine-d3 hydrochloride | Ivabradine D3 Hydrochloride | Others |
Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. Ivabradine D3 Hydrochloride is the deuterium labeled Ivabradine hydrochloride. | |||
T37160 | 8-Demethyl Ivabradine | ||
8-Demethyl Ivabradine is a metabolite derived from Ivabradine, an orally bioavailable cyclic nucleotide-gated (HCN) channel blocker with hyperpolarization-activated properties[1]. | |||
T11695 | N-Demethyl ivabradine hydrochloride | Ivabradine metabolite N-Demethyl Ivabradine hydrochloride | Others |
N-Demethyl Ivabradine Hcl is a specific inhibitor of the funny channel.N-Demethyl Ivabradine Hcl is a metabolite of Ivabradine. | |||
T11694 | Ivabradine-d6 hydrochloride | Ivabradine D6 hydrochloride | Others |
Ivabradine hydrochloride is a new If inhibitor with IC50 of 2.9 μM, and used as a pure heart rate lowering agent. Ivabradine D6 hydrochloride is the deuterium labeled Ivabradine hydrochloride. | |||
T19447 | N-Demethyl Ivabradine D6 Hydrochloride | Others | |
N-Demethyl Ivabradine D6 Hydrochloride salt is the deuterium labeled N-Demethyl Ivabradine, which is a Ivabradine metabolite. | |||
T73975 | Ivabradine impurity 1 | ||
Ivabradine Impurity 1, identified as an impurity of Ivabradine, is an orally bioavailable compound that functions as a blocker of the hyperpolarization-activated, cyclic nucleotide-gated (HCN) channel [1]. | |||
T73976 | Ivabradine impurity 2 | ||
Ivabradine Impurity 2, an impurity of Ivabradine, is a compound known for its oral bioavailability and mechanism as a blocker of hyperpolarization-activated, cyclic nucleotide-gated (HCN) channels [1]. |