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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T4986 | Imidafenacin | KRP-197,ONO-8025 | AChR |
Imidafenacin (KRP-197)(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM. | |||
T36662 | Imidafenacin Metabolite M4 | Imidafenacin Metabolite M4 | |
Imidafenacin metabolite M4 is a metabolite of the muscarinic acetylcholine receptor antagonist imidafenacin.1It is formed from imidafenacin by the cytochrome P450 (CYP) isoform CYP3A4. 1.Kanayama, N., Kanari, C., Masuda,... |