1
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15399 | GNE-207 | Epigenetic Reader Domain | |
GNE-207 is a selective and orally bioavailable inhibitor of the bromodomain of CBP (IC50: 1 nM). It has a selective index of >2500-fold against BRD4 (1). GNE-207 displays excellent CBP potency (EC50: 18 nM for MYC expres... |