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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T38827 | EZH2-IN-5 | EZH2-IN-5 | |
EZH2-IN-5 is a highly effective inhibitor of EZH2, displaying remarkable potency against both wild-type and mutant Tyr641 EZH2, with IC50 values of 1.52 nM and 4.07 nM, respectively. | |||
T62896 | EZH2-IN-12 | ||
EZH2-IN-12 (Compound 5) is a potent inhibitor of EZH2, which has potential for studies of CNS malignancies. | |||
T39497 | EZH2-IN-4 | EZH2-IN-4 | |
EZH2-IN-4 is a highly potent EZH2 inhibitor that can be taken orally. It exhibits inhibitory effects against wild type (WT) 5-membered (5-mer) EZH2 and mutant 5-mer EZH2, with IC 50 values of 0.923 nM and 2.65 nM, respec... |