2
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T6457 | CTEP | mGluR5 inhibitor,RO 4956371 | GluR |
CTEP (RO 4956371) (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold selectivity over other mGlu receptors. | |||
T12717 | Basimglurant | CTEP Derivative,RG7090 | GluR |
Basimglurant (CTEP Derivative) is a potent, selective and orally available modulator of mGlu5 negative allosteric(Kd of 1.1 nM). |