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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T37201 | CAY10787 | ||
CAY10787 is an oxysterol and a negative allosteric modulator of GABAAreceptors.1,2It reduces GABA-induced currents in HEK cells expressing α1β1γ2or α4β3γ2subunit-containing GABAAreceptors (IC50s = 1.5 and 1 μM, respectiv... |