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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T1972 | GSK-5959 | Epigenetic Reader Domain | |
GSK-5959 is an effective, specific and cell permeable BRPF1 bromodomain inhibitor (IC50: ~80 nM). The selectivity of GSK-5959 for BRPF1 is >100-fold over a panel of 35 other bromodomains, including BRPF2/3 and BET family... | |||
T69752 | BRD1991 | ||
BRD1991 is a chemical compound that specifically disrupts the interaction between Beclin 1 and Bcl-2, thereby inducing autophagy. It accomplishes this without initiating apoptosis or other forms of cell death. | |||
T26896 | BRD1652 | BRD-1652,BRD 1652 | |
BRD1652 is a highly selective and potent GSK3 inhibitor. | |||
TQ0083 | NI-57 | Epigenetic Reader Domain | |
NI-57 is an inhibitor of proteins of bromodomain and plant homeodomain finger-containing (BRPF) family, with IC50s of 3.1, 46 and 140 nM for BRPF1, BRPF2 (BRD1) and BRPF3, respectively. | |||
T1854 | MS436 | Epigenetic Reader Domain | |
MS436 is a selective, small-molecule inhibitor for the BRD4 bromodomains. |