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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T1242 | Alvimopan | Opioid Receptor | |
Alvimopan (LY 246736) is a synthetic trans-3, 4-dimethyl-4-(3-hydroxyphenyl) piperidine with peripherally selective opioid mu receptor antagonist activity. Alvimopan is a selective and competitive antagonist at mu-opioid... | |||
T1242L | Alvimopan monohydrate | ||
Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain. | |||
T22238 | Alvimopan dihydrate (LY246736 dihydrate) | ||
Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC 50 of 1.7 nM. Alvimopan dihydrate is highly selective for μ-opioid receptor ( Ki =0... | |||
T20081 | ADL-08-0011 | ADL 08-0011 | |
ADL-08-0011 is an metabolite of alvimopan. | |||
T70267 | ADL 08-0011 HCl | ||
ADL 08-0011 is an active metabolite of the μ-opioid receptor antagonist alvimopan. It is produced from alvimopan via amide hydrolysis by gut microbiota. ADL 08-0011 is a μ-opioid receptor antagonist (Ki = 0.25 nM). It is... |