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Search Result

Search Results for " a1a "

9

Compounds

3

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T60580 A1AR antagonist 2
A1AR antagonist 2 (compound 18h) is a potent antagonist of the A1 adenosine receptor (AR). A1AR antagonist 2 has Ki values of 1.49, 10.2, and 50.1 nM for hA 1, hA 2A, and hA 2B, respectively [1].
T60687 A1AR antagonist 1
A1AR antagonist 1 (compound 18g) is a potent antagonist of A1 adenosine receptor (AR). A1AR antagonist 1 has Ki values of 2.08, 6.91, and 31.2 nM for hA1, hA2A and hA2B, respectively [1].
T61536 A1AR antagonist 4
A1AR antagonist 4 (compound 22) is a highly developed chemical compound that acts as a potent and selective antagonist of the A1 adenosine receptor (A1AR). It possesses a pIC50 value of 5.51 and a pKi value of 6.29 [1].
T72661 A1AT modulator 2
A1AT Modulator 2, an α-1 antitrypsin (A1AT) modulator, exhibits an IC50 value greater than 1.0 μM and an EC50 value less than 0.4 μM. It is utilized in the study of infection and inflammation.
T60615 A1AR antagonist 6
A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].
T62348 A1AR antagonist 3
A1AR antagonist 3 (compound 13) is a selective adenylate 1 (A1) receptor antagonist that acts on human A1 (Ki: 9.69 nM) and rat A1 (Ki: 0.529 nM). A1AR antagonist 3 can be used to study neurological diseases.
T60915 A1AR antagonist 5
A1AR antagonist 5 (compound 20) is a potent and selective antagonist of A1 adenosine receptor (A1AR) with a pKi of 6.11 and a pIC 50 of 5.83 [1].
T83227 A1AT modulator 1
A1AT Modulator 1 potently inhibits Z α1-antitrypsin (A1AT) polymerization, exhibiting a pIC50 of 8.3 [1].
T27509 GW-493838 GW 493838X,GW 493838,GW493838,GW493838X,GW-493838X Adenosine Receptor
GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia or peripheral nerve damage caused by trauma or surgery.

Recombinant Proteins

Species：
Human (2)
Mouse (1)
Expression System：
HEK293 (1)
Human Cells (1)
in vitro E. coli expression system (1)
Tag：
C-6His (1)
His (1)
N-terminal 10xHis-tagged (1)
Cat No. Product Name Species Expression System
TMPJ-00452 Serpin A1a Protein, Mouse, Recombinant (His) Mouse Human Cells
Serpin A1a is also known as alpha-1-antitrypsin, is a member of the serpin superfamily of serine proteinase inhibitors that are involved in the regulation of a number of proteolytic processes. Its primary target is elast...
TMPY-00915 Serpin A1 Protein, Human, Recombinant (His) Human HEK293
SerpinA1, also known as Alpha-1 antitrypsin (AAT), is a prototype member of the Serpin superfamily of the serine protease inhibitors. This serine protease inhibitor blocks the protease, neutrophil elastase. Alpha-1 antit...
TMPH-00892 A1AR Protein, Human, Recombinant (His) Human in vitro E. coli expression system
Receptor for adenosine. The activity of this receptor is mediated by G proteins which inhibit adenylyl cyclase.
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