2
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
TP2048L | α-helical CRF 9-41 acetate | α-helical CRF 9-41 acetate(90880-23-2 Free base) | CRFR |
α-helical CRF 9-41 acetate is a competitive antagonist of CRF2 (KB = 100 nM) and a partial agonist of CRF1 (EC50 = 140 nM). | |||
TP2048 | α-Helical CRF(9-41) | α-helical CRF 9-41 | |
Corticotropin-releasing factor receptor antagonist (Ki values are 17, 5 and 0.97 at human CRF1, rat CRF2α and mouse CRF2β receptors respectively). |