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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12639 | (R)-PS210 | Others | |
(R)-PS210, the R enantiomer of PS210 is a substrate-selective allosteric PDK1 activator with an (AC50 of 1.8 μM). | |||
T16670 | PS210 | PDK | |
PS210 is a potent and selective activator of PDK1 (Kd: 3 μM), specifically targeting the PIF-binding pocket of PDK1, without acting against other protein kinases such as S6K, PKB/Akt, or GSK3. Its prodrug, PS423, serves ... |