Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Compound 40, NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal), a macrocyclic analogue of Ape13, acts as a potent APJ agonist with a Ki of 5.7 nM. It demonstrates favorable Gα12-biased signaling and possesses an enhanced in vivo half-life [1].
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Description | Compound 40, NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal), a macrocyclic analogue of Ape13, acts as a potent APJ agonist with a Ki of 5.7 nM. It demonstrates favorable Gα12-biased signaling and possesses an enhanced in vivo half-life [1]. |
Molecular Weight | 1020.18 |
Formula | C49H73N13O11 |
CAS No. | 2891469-81-9 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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NH2-c[X-R-L-S-X]-K-G-P-(D-2Nal) 2891469-81-9 Others inhibitor inhibit