1
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T17066 | Umbralisib hydrochloride | RP5264 hydrochloride , TGR-1202 hydrochloride | PI3K |
Umbralisib hydrochloride is a novel PI3Kδ inhibitor (IC50 and EC50 of 22.2 nM and 24.3 nM, respectively). Umbralisib hydrochloride is also active against CK1ε (EC50: 6.0 μM). |