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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T15240 | Tazemetostat trihydrochloride | EPZ-6438 trihydrochloride , E-7438 trihydrochloride | Histone Methyltransferase |
Tazemetostat trihydrochloride is a selective and orally available inhibitor of EZH2 (IC50: 4 nM for rat EZH2). It inhibits the activity of human PRC2-containing wild-type EZH2 (Ki: 2.5 nM). It inhibits EZH2 (IC50s: 11 an... |