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TG4-155

Catalog No. T5482    CAS 1164462-05-8   

TG4-155 is a brain penetrant EP2 antagonist (KB = 2.4 nM) that is over 1000-fold less effective at EP4 (KB = 11.4 μM) and a panel of other receptors and channels

Pack Size Availability Price/USD Quantity
2 mg In stock 63.00
5 mg In stock 89.00
10 mg In stock 151.00
25 mg In stock 306.00
50 mg In stock 533.00
100 mg In stock 800.00
1 mL * 10 mM (in DMSO) In stock 98.00
Bulk Size: Please Quote for Discount Please Quote for Bulk Size
Biological Activity:

Product Description:

TG4-155 is a brain penetrant EP2 antagonist (KB = 2.4 nM) that is over 1000-fold less effective at EP4 (KB = 11.4 μM) and a panel of other receptors and channels

Receptor:

EP2;

Chemical Information:
Molecular Weight 394.47
Formula C23H26N2O4
CAS Number 1164462-05-8
Solubility

DMSO: 125 mg/mL (316.89 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage store at -80°C
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.