Shopping Cart
  • Remove All
  • TargetMol
    Your shopping cart is currently empty
TargetMol | Compound Library

Anti-Cancer Compound Library

Catalog No. L2100

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 9332 compounds with anti-tumor activity based on different characteristics and abnormal metabolism with cancer cells. All of these compounds are the small molecules modulating the metabolism, growth, invasion, and metastasis of tumor cells that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Resource Download
Library compound info
Excel
SDF
Contact us for more batch information

Catalog No. L2100

Anti-Cancer Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
Inquiry & Custom

Top Publication Citing
Use of TargetMol Products

Cite scientific literature on TargetMol products

View More

Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Product Description Product Description

  • A unique collection of 9332 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization | TargetMol Library Customization

Compound Library | TargetMol
Targetmol Compound Libraries
can be highly customized!
Inquiry & Custom

Sci Citations

Library Customization | TargetMol Library Composition

Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Antibacterial
DNA/RNA Synthesis
NF-κB
COX
Adrenergic Receptor
CDK
Dopamine Receptor
PI3K
EGFR
Potassium Channel
Epigenetic Reader Domain
Calcium Channel
Reactive Oxygen Species
Histamine Receptor
VEGFR
Antibiotic
Cytochromes P450
Sodium Channel
Histone Methyltransferase
HDAC
GABA Receptor
TRP/TRPV Channel
JAK
Parasite
mTOR
Akt
PPAR
ERK
Wnt/beta-catenin
HIV Protease
AChR
GPCR
PARP
Antifungal
PKC
Prostaglandin Receptor
Estrogen Receptor/ERR
Src
FLT
STAT
p38 MAPK
FGFR
Microtubule Associated
Adenosine Receptor
AMPK
PDGFR
Topoisomerase
GSK-3
Nucleoside Antimetabolite/Analog
Dehydrogenase
TNF
Estrogen/progestogen Receptor
Opioid Receptor
Caspase
Raf
Glucocorticoid Receptor
Bcl-2 Family
Influenza Virus
Antioxidant
iGluR
c-Met/HGFR
Ferroptosis
Androgen Receptor
c-Kit
HSP
Sirtuin
ALK
Bcr-Abl
Cannabinoid Receptor
ATPase
MMP
Histone Demethylase
Ras
TGF-beta/Smad
Aurora Kinase
IL Receptor
Phosphatase
PDE
ROCK
DUB
JNK
ROS
MAPK
MEK
Tyrosine Kinases
NO Synthase
p53
P-gp
IκB/IKK
Mitophagy
RIP kinase
Lipoxygenase
NMDAR
SARS-CoV
Virus Protease
Serine/threonin kinase
S1P Receptor
HIF/HIF Prolyl-Hydroxylase
CXCR
HSV
PKA
Antiviral
NOD
DNA-PK
Hedgehog/Smoothened
IGF-1R
Nrf2
c-RET
Histone Acetyltransferase
LPL Receptor
TLR
ATM/ATR
Drug Metabolite
P2X Receptor
S6 Kinase
E1/E2/E3 Enzyme
FAK
Casein Kinase
HER
HIF
Cholinesterase (ChE)
PERK
PLK
Mitochondrial Metabolism
Pim
Sigma receptor
TAM Receptor
Chk
Chloride channel
DNA Methyltransferase
Interleukin
Neurokinin receptor
NOS
Proteasome
GluR
RAAS
Serotonin Transporter
Beta Amyloid
Gamma-secretase
HBV
HCV Protease
Norepinephrine
Phospholipase
Rho
Tyrosinase
DHFR
DNA Alkylator/Crosslinker
Protease-activated Receptor
Proton pump
Trk receptor
Endothelin Receptor
Mdm2
Carbonic Anhydrase
Glucagon Receptor
IRAK
MAO
PDK
PROTACs
DYRK
Retinoid Receptor
SGLT
Syk
Antifection
Fatty Acid Synthase
P2Y Receptor
PD-1/PD-L1
Smo
c-Fms
c-Myc
DNA
Guanylate cyclase
Neuropeptide Y Receptor
Reverse Transcriptase
transporter
Kras
CaMK
cAMP
CFTR
LPA Receptor
Transferase
Anti-infection
DNA Alkylation
Integrin
IRE1
OX Receptor
ROS Kinase
ADC Cytotoxin
Cholecystokinin Receptor
HMG-CoA Reductase
Leukotriene Receptor
NADPH
ABC Transporter
Antifolate
IAP
Kinesin
Monoamine Oxidase
PI4K
Progesterone Receptor
Serine Protease
Vasopressin Receptor
YAP
GTPase
MRP
NOD-like Receptor (NLR)
GHSR
Indoleamine 2,3-Dioxygenase (IDO)
MicroRNA
BTK
Aromatase
CSF-1R
GPCR19
Monocarboxylate transporter
Reductase
Bradykinin Receptor
CCR
GRK
Immunology/Inflammation related
Ligand for E3 Ligase
Neurotensin Receptor
Somatostatin
AhR
Aryl Hydrocarbon Receptor
Glutathione Peroxidase
Melanocortin Receptor
Melatonin Receptor
Telomerase
BCRP
Free radical scavengers
FXR
Glucosidase
LIM Kinase
MNK
Monoamine Transporter
Myosin
PAD
STING
CaSR
Ephrin Receptor
GNRH Receptor
IFNAR
LTR
Na+/Ca2+ Exchanger
PAK
PGE Synthase
PTEN
SIK
Thrombin
Wee1
Acyltransferase
APC/C
Arrestin
BACE
Bombesin Receptor
Glucokinase
Glutaminase
GPX
Hydroxylase
Isocitrate Dehydrogenase (IDH)
LDL
Liver X Receptor
Methionine Adenosyltransferase (MAT)
MLK
Molecular Glues
OCT
Tie-2
UGT
Amino Acids and Derivatives
Annexin A
CRFR
CRM1
Cysteine Protease
Ligands for Target Protein for PROTAC
Lipid
LRRK2
Melanin-concentrating Hormone Receptor (MCHR)
MELK
MT Receptor
NAMPT
OAT
PAFR
PYK2
ribosome
RSV
SGK
Survivin
ACK1
Apelin receptor
ASK
Beta-Secretase
BMI-1
Carboxypeptidase
Cell Cycle Arrest
CGRP Receptor
CRISPR/Cas9
Discoidin Domain Receptor (DDR)
DPP-4
FAAH
MTH1
NPC1L1
Oxytocin Receptor
PKM
Platelet aggregation
Porcupine
ROR
TOPK
Xanthine Oxidase
Adenosine Deaminase
Adiponectin Receptor
Aminopeptidase
Aquaporin
ATP Citrate Lyase
Decarboxylase
DNA gyrase
GST
Hck
Hexokinase
Hippo pathway
IDO
MALT
p97
PAI-1
Pyroptosis
RANKL/RANK
TSH Receptor
AAK1
CD73
Complement System
DAPK
Factor Xa
Haspin Kinase
HCN Channel
HuR
Imidazoline Receptor
KLF
KSP
Na-K-Cl cotransporter
NEDD8
RAR/RXR
VDAC
Adenylyl Cyclase
AIM2
Arginase
Cell wall
EBI2/GPR183
Epoxide Hydrolase
Galectin
Gap Junction Protein
GluCls
Glutathione reductase
gp120/CD4
Lipase
Lysosomal Autophagy
MyD88
NADPH-oxidase
OXPHOS
Protease
PSMA
RXFP receptor
Thrombopoietin Receptor
VDA
FOXO3
IKZF
Vitamin
Advanced Glycation End Products
Amylase
Angiotensin-converting Enzyme (ACE)
Anion Exchanger
CD38
cGAS
CYP19A1
Dynamin
Endonuclease
FLAP
Glyoxalase
GlyT
hCE
Huntingtin
Hydrogenase
N-Acetylglucosaminyltransferase
Necroptosis
NEDD4-1
Neprilysin
Neuropeptide W
NUDIX hydrolase
Phosphorylase
Piezo Channel
PROTAC Linker
Stearoyl-CoA Desaturase (SCD)
Stemness kinase
Thioredoxin
Transaminase
Transketolase
Sodium-dependent phosphate transporter

Keywords