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TargetMol | Compound Library

Anti-Cancer Compound Library

Catalog No. L2100

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy, however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients). We carefully select 9332 compounds with anti-tumor activity based on different characteristics and abnormal metabolism with cancer cells. All of these compounds are the small molecules modulating the metabolism, growth, invasion, and metastasis of tumor cells that can be used for tumor-related research and anti-tumor drug screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2100

Anti-Cancer Compound Library

sizeIn stock

  • 1 mg
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Product Description Product Description

  • A unique collection of 9332 compounds with anti-cancer activity for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity and safety profiled in (confirmed by) pre-clinical and clinical settings (research and trials);
  • Effective tool for molecular mechanism of tumorigenesis, and anti-tumor drug screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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Apoptosis
Autophagy
5-HT Receptor
Endogenous Metabolite
Antibacterial
NF-κB
DNA/RNA Synthesis
COX
Adrenergic Receptor
CDK
Dopamine Receptor
PI3K
EGFR
Potassium Channel
Epigenetic Reader Domain
Reactive Oxygen Species
Antibiotic
Calcium Channel
Histamine Receptor
VEGFR
Cytochromes P450
Sodium Channel
Histone Methyltransferase
HDAC
GABA Receptor
Parasite
TRP/TRPV Channel
JAK
PPAR
Akt
mTOR
ERK
Wnt/beta-catenin
AChR
HIV Protease
Antifungal
GPCR
PARP
PKC
Prostaglandin Receptor
Estrogen Receptor/ERR
Src
FLT
STAT
p38 MAPK
FGFR
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Adenosine Receptor
AMPK
PDGFR
GSK-3
Nucleoside Antimetabolite/Analog
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TNF
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Influenza Virus
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ALK
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ATPase
MMP
Histone Demethylase
Ras
TGF-beta/Smad
Aurora Kinase
IL Receptor
Phosphatase
PDE
ROCK
DUB
JNK
ROS
MAPK
MEK
P-gp
Tyrosine Kinases
NO Synthase
p53
IκB/IKK
Mitophagy
RIP kinase
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Lipoxygenase
NMDAR
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S1P Receptor
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IGF-1R
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LPL Receptor
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P2X Receptor
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FAK
Casein Kinase
HER
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PERK
PLK
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Pim
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transporter
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IRE1
OX Receptor
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ABC Transporter
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Progesterone Receptor
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Neurotensin Receptor
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STING
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Ligands for Target Protein for PROTAC
Lipid
LRRK2
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MELK
MT Receptor
NAMPT
OAT
PAFR
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ribosome
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ASK
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Oxytocin Receptor
PKM
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TOPK
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Adiponectin Receptor
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Piezo Channel
PROTAC Linker
Stearoyl-CoA Desaturase (SCD)
Stemness kinase
Thioredoxin
Transaminase
Transketolase
Sodium-dependent phosphate transporter
Vitamin

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