Powder: -20°C for 3 years | In solvent: -80°C for 1 year
SCH442416 (SCH 442416) is an selective antagonist of adenosine A2A receptor. SCH442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 40.00 | |
2 mg | In stock | $ 57.00 | |
5 mg | In stock | $ 85.00 | |
10 mg | In stock | $ 142.00 | |
25 mg | In stock | $ 296.00 | |
50 mg | In stock | $ 473.00 | |
100 mg | In stock | $ 693.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 98.00 |
Description | SCH442416 (SCH 442416) is an selective antagonist of adenosine A2A receptor. SCH442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.048 and 0.5 nM respectively). |
Targets&IC50 | A2AR (rat):0.5 nM (IC50), A2AR (human):0.048 nM (IC50) |
In vitro | The A2A receptor antagonist (SCH 442416) could increase mRNA expression of the Kir 2.1and Kir 4.1 channels in Müller cells to protect the retinal neurons in vitro under hypoxic conditions[1]. |
Synonyms | SCH 442416 |
Molecular Weight | 389.41 |
Formula | C20H19N7O2 |
CAS No. | 316173-57-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 60 mg/ml (154.08 mM)
You can also refer to dose conversion for different animals. More
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SCH442416 316173-57-6 GPCR/G Protein Neuroscience Adenosine Receptor SCH-442416 A2A imaging inhibit P1 receptor Inhibitor SCH 442416 adenosine inhibitor