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Relebactam

Catalog No. T4017 CAS 1174018-99-5

Synonyms: MK-7655

Relebactam (MK-7655) is a diazabicyclooctane inhibitor with activity against a wide spectrum of β-lactamases.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

Relebactam, CAS 1174018-99-5

Pack Size	Availability	Price/USD
1 mg	In stock	$ 44.00
5 mg	In stock	$ 97.00
10 mg	In stock	$ 155.00
25 mg	In stock	$ 289.00
50 mg	In stock	$ 538.00
100 mg	In stock	$ 778.00
1 mL * 10 mM (in DMSO)	In stock	$ 113.00

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Purity: 100%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Relebactam (MK-7655) is a diazabicyclooctane inhibitor with activity against a wide spectrum of β-lactamases.

Synonyms	MK-7655
Molecular Weight	348.38
Formula	C12H20N4O6S
CAS No.	1174018-99-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 3.48 mg/mL (10 mM), Sonication is recommended.

References and Literature

1. Lapuebla A, et al. Activity of Imipenem with Relebactam against Gram-Negative Pathogens from New York City. Antimicrob Agents Chemother. 2015 Aug;59(8):5029-31. 2. Bush K., et al. A resurgence of β-lactamase inhibitor combinations effective against multidrug-resistant Gram-negative pathogens. Int J Antimicrob Agents. 2015 Nov;46(5):483-93.

Related compound libraries

This product is contained In the following compound libraries：

EMA Approved Drug Library Inhibitor Library Drug Repurposing Compound Library Beta-Lactam Compound Library Human Metabolite Library Drug-induced Liver Injury (DILI) Compound Library Antibiotics Library Pediatric Drug Library Anti-Bacterial Compound Library Approved Drug Library

Related Products

Related compounds with same targets

Chlorquinaldol GSK2200150A Clorophene 7-Aminocephalosporanic acid Diniconazole Sodium citrate dihydrate S-Methyl methanesulfonothioate Patchouli alcohol

Dose Conversion

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Calculation results:

Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

Note:

Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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An example of a molarity calculation using the molarity calculator
What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
Enter 197.13 into the Molecular Weight (MW) box
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The answer of 19.713 mg appears in the Mass box

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The dilution calculator is a useful tool which allows you to calculate how to dilute a stock solution of known concentration. Enter C1, C2 & V2 to calculate V1.

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An example of a dilution calculation using the Tocris dilution calculator
What volume of a given 10 mM stock solution is required to make 20ml of a 50 μM solution?
Using the equation C1V1 = C2V2, where C1=10 mM, C2=50 μM, V2=20 ml and V1 is the unknown:
Enter 10 into the Concentration (start) box and select the correct unit (millimolar)
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The answer of 100 microliter (0.1 ml) appears in the Volume (start) box

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Molecule Formula

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Definitions of molecular mass, molecular weight, molar mass and molar weight:
Molecular mass (molecular weight) is the mass of one molecule of a substance and is expressed n the unified atomic mass units (u). (1 u is equal to 1/12 the mass of one atom of carbon-12)
Molar mass (molar weight) is the mass of one mole of a substance and is expressed in g/mol.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Relebactam 1174018-99-5 Microbiology/Virology Antibacterial antibacterial Inhibitor P. aeruginosa inhibit Imipenem β-lactamases MK 7655 Bacterial Enterobacteriaceae MK7655 MK-7655 inhibitor

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.