Powder: -20°C for 3 years | In solvent: -80°C for 1 year
RP-001 is a selective agonist of picomolar short-acting S1P1 (EDG1)(EC50 of 9 pM), has little activity on S1P2-S1P4 and only moderate affinity for S1P5.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 8-10 weeks | $ 2,120.00 | |
50 mg | 8-10 weeks | $ 2,780.00 | |
100 mg | 8-10 weeks | $ 3,700.00 |
Description | RP-001 is a selective agonist of picomolar short-acting S1P1 (EDG1)(EC50 of 9 pM), has little activity on S1P2-S1P4 and only moderate affinity for S1P5. |
In vitro | dose-dependent lymphopenia of CD4+ T cells elicited by RP-001. RP-001 induces acute lymphopenia with rapid recovery to untreated levels. |
In vivo | Dose-dependent rapid lymphopenia caused by RP-001 (EC50 of 0.03 mg/kg). |
Molecular Weight | 432.47 |
Formula | C24H24N4O4 |
CAS No. | 1306761-53-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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RP-001 1306761-53-4 Others RP001 RP 001 inhibitor inhibit