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PKG inhibitor peptide

Catalog No. TP1903 CAS 82801-73-8

Synonyms: cGMP Dependent Kinase Inhibitor Peptide

Competitive inhibitor of cGMP-dependent protein kinase (PKG); analog of a substrate peptide corresponding to a phosphorylation site of histone H2B. Competes with synthetic substrates (Ki = 86 mM) but does not inhibit phosphorylation of intact histones by PKG. Inhibits phosphorylation of intact histones by PKA.

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PKG inhibitor peptide Chemical Structure

PKG inhibitor peptide, CAS 82801-73-8

Pack Size	Availability	Price/USD	Quantity
1 mg	35 days	$ 143.00
5 mg	35 days	$ 655.00

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Biological Description

Chemical Properties

Storage & Solubility Information

Description

Synonyms	cGMP Dependent Kinase Inhibitor Peptide
Molecular Weight	943.12
Formula	C38H74N18O10
CAS No.	82801-73-8

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Bhatnagar et al (1988) Synthetic peptide analogues differentially alter the binding affinities of cyclic nucleotide dependent protein kinases for nucleotide substrates. Biochemistry 27 1988 PMID: 2. Glass (1983) Differential responses of cyclic GMP-dependent and cyclic AMP-dependent protein kinases to synthetic peptide inhibitors. Biochem.J. 213 159 PMID: 3. Glass et al (1986) Differential and common recognition of the catalytic sites of the cGMP-dependent and cAMP-dependent protein kinases by inhibitory peptides derived from the heat-stable inhibitor protein. J.Biol.Chem. 261 12166 PMID:

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

PKG inhibitor peptide 82801-73-8 cGMP Dependent Kinase Inhibitor Peptide inhibitor inhibit

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.