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PGlu-3-methyl-His-Pro-NH2 TFA

Catalog No. T19511 CAS T19511

Synonyms: A-42872 TFA

PGlu-3-methyl-His-Pro-NH2 TFA, enhances binding to pituitary TRH receptors and increases stimulation of thyroid-stimulating hormone (TSH) release from the pituitary.

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PGlu-3-methyl-His-Pro-NH2 TFA Chemical Structure

PGlu-3-methyl-His-Pro-NH2 TFA, CAS T19511

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Biological Description

Chemical Properties

Storage & Solubility Information

Description	PGlu-3-methyl-His-Pro-NH2 TFA, enhances binding to pituitary TRH receptors and increases stimulation of thyroid-stimulating hormone (TSH) release from the pituitary.
In vitro	PGlu-3-methyl-His-Pro-NH2 TFA is more potent in eliciting behavioral effects as well as being more potent in the release of both growth hormone and thyroid stimulating hormone[1].

Synonyms	A-42872 TFA
Molecular Weight	490.43
Formula	C19H25F3N6O6
CAS No.	T19511

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

H2O: 250 mg/mL (509.76 mM), Sonication is recommended.

References and Literature

1. Koskinen LO, et al. Cerebrovascular effects of the TRH analogues pGlu-3-methyl-His-Pro amide and pGlu-Glu-Pro amide: a comparison with TRH. Ups J Med Sci. 2000;105(1):73-83. 2. Magnusson BM, et al. Biological effects after percutaneous absorption of thyrotropin-releasing hormone and its analogue M-TRH. Peptides. 2001 Jan;22(1):73-9.

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Keywords

PGlu-3-methyl-His-Pro-NH2 TFA T19511 Others PGlu-3-methyl-His-Pro-NH-2 TFA PGlu 3 methyl His Pro NH2 TFA PGlu3methylHisProNH2 TFA A-42872 TFA inhibitor inhibit

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