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Org 25543

Catalog No. T50082 CAS 363628-88-0

Org 25543 is the development of an N-Acyl amino acid that selectively inhibits the glycine <a href="/target/transporter" style="display: inline; color: #c13a36">transporter</a> 2 to produce analgesia in a rat model of chronic pain.

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Org 25543, CAS 363628-88-0

Pack Size	Availability	Price/USD
1 mg	In stock	$ 127.00
2 mg	In stock	$ 189.00
5 mg	In stock	$ 293.00
10 mg	In stock	$ 439.00
25 mg	In stock	$ 751.00
50 mg	In stock	$ 1,125.00
100 mg	In stock	$ 1,688.00

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Purity: 99.13%

Biological Description

Chemical Properties

Storage & Solubility Information

Description

Org 25543 is the development of an N-Acyl amino acid that selectively inhibits the glycine transporter 2 to produce analgesia in a rat model of chronic pain.

Molecular Weight	412.53
Formula	C24H32N2O4
CAS No.	363628-88-0

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Mostyn SN, et al. Development of an N-Acyl Amino Acid That Selectively Inhibits the Glycine Transporter 2 To Produce Analgesia in a Rat Model of Chronic Pain. J Med Chem. 2019 Mar 14;62(5):2466-2484.

Related compound libraries

This product is contained In the following compound libraries：

Bioactive Compound Library Ion Channel Inhibitor Library Anti-Cancer Compound Library Bioactive Compounds Library Max NO PAINS Compound Library

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Keywords

Org 25543 363628-88-0 Membrane transporter/Ion channel Chloride channel Inhibitor inhibitor inhibit

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