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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10829 | CKI-7 free base | CKI-7 | Casein Kinase |
CKI-7 free base is a potent and ATP-competitive inhibitor of casein kinase 1 (CK1; IC50: 6 μM; Ki: 8.5 μM) and a selective Cdc7 kinase inhibitor. CKI-7 free base also inhibits SGK, ribosomal S6 kinase-1 (S6K1), and MSK1. |