Powder: -20°C for 3 years | In solvent: -80°C for 1 year
CBB1007 Hcl is a selective, reversible, and substrate competitive LSD1 inhibitor (IC50: 5.27 μM for hLSD1).
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
2 mg | Inquiry | $ 140.00 | |
5 mg | Inquiry | $ 207.00 | |
10 mg | Inquiry | $ 314.00 | |
50 mg | Inquiry | $ 739.00 | |
100 mg | Inquiry | $ 1,148.00 | |
200 mg | Inquiry | Inquiry | |
500 mg | Inquiry | Inquiry |
Description | CBB1007 Hcl is a selective, reversible, and substrate competitive LSD1 inhibitor (IC50: 5.27 μM for hLSD1). |
In vitro | CBB1007 efficiently can block LSD1-mediated demethylation of H3K4Me2 and H3K4Me (IC50 ≤ 5 μM) with no effect on H3K4Me3 and H3K9Me2, and LSD2 and JARID1A activities. Increases H3K4Me2 and H3K4Me contents (IC50 ≤ 5 μM), and causes activation of epigenetically suppressed CHRM4/M4-ArchR and SCN3A genes in F9 cells (IC50 ≤ 3.74 μM). |
Synonyms | CBB1007 hydrochloride |
Molecular Weight | 716.91 |
Formula | C27H39Cl5N8O4 |
CAS No. | T10699 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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CBB1007 hydrochloride (1379573-92-8 free base) T10699 Others 1379573-92-8 free base CBB-1007 Hydrochloride CBB-1007 hydrochloride (1379573-92-8 free base) CBB1007 hydrochloride (1379573928 free base) CBB 1007 Hydrochloride 1379573-92-8 CBB1007 Hydrochloride CBB1007 hydrochloride (1379573 92 8 free base) CBB1007 hydrochloride inhibitor inhibit