Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Capsaicin is the primary active component of the heat and pain-eliciting lipid soluble fraction of the Capsicum pepper. Capsaicin signals are transduced by a heat-activated ion channel, the vanilloid receptor 1 (VR1), or transient receptor potential vanilloid 1 (TRPV1). CAY10448 is an iodinated nonivamide, a potent capsaicin receptor antagonist with an IC50 value of approximately 10 nM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | 35 days | $ 53.00 | |
5 mg | 35 days | $ 223.00 | |
10 mg | 35 days | $ 393.00 | |
50 mg | 35 days | $ 1,700.00 |
Description | Capsaicin is the primary active component of the heat and pain-eliciting lipid soluble fraction of the Capsicum pepper. Capsaicin signals are transduced by a heat-activated ion channel, the vanilloid receptor 1 (VR1), or transient receptor potential vanilloid 1 (TRPV1). CAY10448 is an iodinated nonivamide, a potent capsaicin receptor antagonist with an IC50 value of approximately 10 nM. |
Synonyms | CAY10448 |
Molecular Weight | 433.32 |
Formula | C18H28INO3 |
CAS No. | 1177195-52-6 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Ethanol: 30 mg/mL
Ethanol:PBS (pH 7.2)(1:2): 0.25 mg/mL
DMF: 30 mg/mL
DMSO: 30 mg/mL
You can also refer to dose conversion for different animals. More
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CAY10448 1177195-52-6 CAY 10448 CAY-10448 inhibitor inhibit