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Bremelanotide Acetate

Catalog No. T7608   CAS 1607799-13-2
Synonyms: bremelanotide, PT-141 Acetate

Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .

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Bremelanotide Acetate Chemical Structure
Bremelanotide Acetate, CAS 1607799-13-2
Pack Size Availability Price/USD Quantity
10 mg In stock $ 46.00
25 mg In stock $ 83.00
50 mg In stock $ 139.00
100 mg In stock $ 207.00
1 mL * 10 mM (in DMSO) In stock $ 65.00
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Purity: 98%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description Bremelanotide Acetate (PT-141 Acetate) is an agonist of melanocortin receptor (MCR) .
In vivo Treatment with Bremelanotide?(100 or 200 μg/kg) significantly increased proceptive solicitations in females primed with E+Por E alone (E+O) in bilevel chambers[1]
Animal Research Bremelanotide(PT-141), a cyclic heptapeptide melanocortin analogue (Palatin Technologies, Cranbury, NJ), was dissolved in saline to obtain doses of 50, 100, and 200 μg/kg/ml, and injected s.c. 5 min before each behavioral test. An equal volume of saline was administered to control animals[1].
Synonyms bremelanotide, PT-141 Acetate
Molecular Weight 1085.22
Formula C52H72N14O12
CAS No. 1607799-13-2

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 36 mg/mL (33.17 mM)

TargetMolReferences and Literature

1. Pfaus JG, Shadiack A, Van Soest T,et al.Selective facilitation of sexual solicitation in the female rat by a melanocortin receptor agonist[J].Proc Natl Acad Sci U S A. 2004 Jul 6;101(27) 2. Clayton AH, Althof SE, Kingsberg S,et al.Bremelanotide for female sexual dysfunctions in premenopausal women: a randomized, placebo-controlled dose-finding trial[J].Womens Health (Lond). 2016 Jun;12(3):325-37.

Related compound libraries

This product is contained In the following compound libraries:
Peptide Compound Library Anti-Cancer Clinical Compound Library GPCR Compound Library Anti-Cancer Drug Library Anti-Cancer Approved Drug Library Membrane Protein-targeted Compound Library Drug Repurposing Compound Library FDA-Approved Drug Library FDA-Approved & Pharmacopeia Drug Library Bioactive Compounds Library Max

Related Products

Related compounds with same targets
Melanotan (MT)-II N,N′-Diferuloylputrescine Adrenocorticotropic Hormone (ACTH) (4-10), human HS024 Dersimelagon THIQ Setmelanotide SHU 9119 acetate

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Keywords

Bremelanotide Acetate 1607799-13-2 GPCR/G Protein Neuroscience Melanocortin Receptor PT 141 Acetate bremelanotide inhibit PT141 PT141 Acetate PT-141 Acetate MC Receptor PT 141 Inhibitor PT-141 inhibitor

 

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