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Balovaptan

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Purity:99.34%

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COA HNMR HPLC

Balovaptan

Catalog No. T14494Cas No. 1228088-30-9

Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors. It is used for the research of autism.

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Pack Size	Price	Availability
5 mg	$60	In Stock
10 mg	$97	In Stock
25 mg	$197	In Stock
50 mg	$318	In Stock
100 mg	$497	In Stock
1 mL x 10 mM (in DMSO)	$67	In Stock

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Product Introduction

Bioactivity

Description	Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors. It is used for the research of autism.
In vitro	Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for hV1a and mhV1a. It is used for the research of autism. Balovaptan shows >30000-fold selectivity for hV1a over hV2 receptors, 9891-fold selectivity over hOTR (human oxytocin receptor)[1].
Alias	RG7314

Chemical Properties

Molecular Weight	409.91
Formula	C22H24ClN5O
Cas No.	1228088-30-9

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 62.5 mg/mL (152.47 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.4396 mL	12.1978 mL	24.3956 mL	121.9780 mL
5 mM	0.4879 mL	2.4396 mL	4.8791 mL	24.3956 mL
10 mM	0.2440 mL	1.2198 mL	2.4396 mL	12.1978 mL
20 mM	0.1220 mL	0.6099 mL	1.2198 mL	6.0989 mL
50 mM	0.0488 mL	0.2440 mL	0.4879 mL	2.4396 mL
100 mM	0.0244 mL	0.1220 mL	0.2440 mL	1.2198 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

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A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% ddH2O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLddH2O TargetMol | reagent

mix well and clarify

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