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BMS-986020

Catalog No. T4016 CAS 1257213-50-5

Synonyms: AM152, BMS986020, BMS 986020

BMS-986020 is a selective antagonist of LPA1.

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BMS-986020, CAS 1257213-50-5

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Purity: 98%

Biological Description

Chemical Properties

Storage & Solubility Information

Description	BMS-986020 is a selective antagonist of LPA1.
Targets&IC50	MRP4:6.2 µM (IC50), BSEP:4.8 µM (IC50), MDR3:7.5 µM (IC50)

Synonyms	AM152, BMS986020, BMS 986020
Molecular Weight	482.536
Formula	C29H26N2O5
CAS No.	1257213-50-5

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 2 years

Solubility Information

DMSO: 64 mg/mL

( < 1 mg/ml refers to the product slightly soluble or insoluble )

References and Literature

1. Kihara Y et al. Lysophospholipid receptors in drug discovery. Exp Cell Res. 2015 May 1;333(2):171-7.

Related compound libraries

This product is contained In the following compound libraries：

GPCR Compound Library Inhibitor Library Immunology/Inflammation Compound Library Anti-Metabolism Disease Compound Library Drug Repurposing Compound Library Neuronal Signaling Compound Library Anti-Fibrosis Compound Library Bioactive Compound Library Clinical Compound Library

Related Products

Related compounds with same targets

TAK-615 Tetradecyl Phosphonate ONO-7300243 Ki16198 TC LPA5 4 H2L5186303 GRI977143 DBIBB

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Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

BMS-986020 1257213-50-5 G蛋白偶联受体 LPA Receptor LPL Receptor inhibit idiopathic AM-152 Lysophospholipid Receptor AM 152 BMS986020 IPF AM152 fibrosis pulmonary BMS 986020 autoradiography Inhibitor ARG inhibitor

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