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BMS-986020

Name: BMS-986020
Brand: TargetMol
SKU: T4016
Price: 47 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T4016Cas No. 1257213-50-5

Alias BMS986020, AM152

BMS-986020 (AM152) is a selective LPA1 antagonist.

BMS-986020

🥰Excellent

Purity: 98.82%

Catalog No. T4016Alias BMS986020, AM152Cas No. 1257213-50-5

BMS-986020 (AM152) is a selective LPA1 antagonist.

Pack Size	Price	Availability
1 mg	$47	In Stock
5 mg	$76	In Stock
10 mg	$122	In Stock
25 mg	$222	In Stock
50 mg	$372	In Stock
100 mg	$556	In Stock
1 mL x 10 mM (in DMSO)	$81	In Stock

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Batch Information

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Purity:98.82%

Resource Download

COA HNMR LCMS

Product Introduction

Bioactivity

Description	BMS-986020 (AM152) is a selective LPA1 antagonist.
Targets&IC50	MDR3:7.5 µM (IC50), BSEP:4.8 µM (IC50), MRP4:6.2 µM (IC50)
Synonyms	BMS986020, AM152

Chemical Properties

Molecular Weight	482.53
Formula	C₂₉H₂₆N₂O₅
Cas No.	1257213-50-5
Smiles	C[C@@H](OC(=O)Nc1c(C)noc1-c1ccc(cc1)-c1ccc(cc1)C1(CC1)C(O)=O)c1ccccc1
Relative Density.	1.309 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 50 mg/mL (103.62 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0724 mL	10.3621 mL	20.7241 mL	103.6205 mL
5 mM	0.4145 mL	2.0724 mL	4.1448 mL	20.7241 mL
10 mM	0.2072 mL	1.0362 mL	2.0724 mL	10.3621 mL
20 mM	0.1036 mL	0.5181 mL	1.0362 mL	5.1810 mL
50 mM	0.0414 mL	0.2072 mL	0.4145 mL	2.0724 mL
100 mM	0.0207 mL	0.1036 mL	0.2072 mL	1.0362 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc