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Catalog No. T4016   CAS 1257213-50-5
Synonyms: AM152, BMS986020

BMS-986020 (AM152) is a selective antagonist of LPA1.

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BMS-986020 Chemical Structure
BMS-986020, CAS 1257213-50-5
Pack Size Availability Price/USD Quantity
1 mg In stock $ 47.00
5 mg In stock $ 76.00
10 mg In stock $ 122.00
25 mg In stock $ 222.00
50 mg In stock $ 372.00
100 mg In stock $ 556.00
1 mL * 10 mM (in DMSO) In stock $ 81.00
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Purity: 100%
Purity: 98.61%
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Biological Description
Chemical Properties
Storage & Solubility Information
Description BMS-986020 (AM152) is a selective antagonist of LPA1.
Targets&IC50 MDR3:7.5 µM (IC50), MRP4:6.2 µM (IC50), BSEP:4.8 µM (IC50)
Synonyms AM152, BMS986020
Molecular Weight 482.53
Formula C29H26N2O5
CAS No. 1257213-50-5


Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 50 mg/mL (103.62 mM)

TargetMolReferences and Literature

1. Kihara Y et al. Lysophospholipid receptors in drug discovery. Exp Cell Res. 2015 May 1;333(2):171-7.

Related compound libraries

This product is contained In the following compound libraries:
Membrane Protein-targeted Compound Library Anti-Cancer Clinical Compound Library Anti-Cancer Drug Library GPCR Compound Library Drug Repurposing Compound Library Inhibitor Library NO PAINS Compound Library Anti-Metabolism Disease Compound Library Bioactive Compound Library Target-Focused Phenotypic Screening Library

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BMS-986278 Ki16198 GRI977143 DBIBB AM095 LX-1031 Tetradecyl Phosphonate H2L 5765834

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BMS-986020 1257213-50-5 GPCR/G Protein LPL Receptor LPA Receptor inhibit idiopathic AM 152 Lysophospholipid Receptor AM152 BMS986020 IPF fibrosis pulmonary AM-152 autoradiography BMS 986020 Inhibitor ARG inhibitor