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TargetMol | Compound Library

Anti-Cancer Clinical Compound Library

Catalog No. L2120

During the past decades, we have witnessed many landmark discoveries and successes in cancer research and therapy,however, cancer is still a major health problem for human beings, and it often physically and emotionally brings pains and difficulties to those living with it. Cancer cells remain undifferentiated (continue to divide, causing more damage, and invading new tissue), lack normal cell signaling responses (loss of contact inhibition and evasion of programmed cell death), contain abnormal changes (genetic abnormalities) in chromatin, have altered energy metabolism, and induce vascularization (ensure a steady supply of oxygen and nutrients).

We carefully select 2760 anti-cancer compounds currently in clinical trial phases based on published literatures and database to form this collection that can be used for high throughput screening and high content screening.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.

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Catalog No. L2120

Anti-Cancer Clinical Compound Library

sizeIn stock

  • 1 mg
  • 10 μL x 10 mM (in DMSO)
  • 20 μL x 10 mM (in DMSO)
  • 30 μL x 10 mM (in DMSO)
  • 50 μL x 10 mM (in DMSO)
  • 100 μL x 10 mM (in DMSO)
  • 250 μL x 10 mM (in DMSO)
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Packaging And Storage Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
  • This compound library is provided at a concentration of 10 mM in DMSO. A small number of compounds may be provided in different solvents or concentrations due to solubility or stability requirements. Please refer to the specific product information for details.

Product Description Product Description

  • A unique collection of 2760 anti-cancer compounds for high throughput screening (HTS) and high content screening (HCS);
  • Bioactivity confirmed by pre-clinical research and all of them are currently in clinical trial phases, representing the cutting-edge treatments for cancers;
  • Effective tool for cancer research and drug repurposing screening;
  • Covers various major targets including PI3K, HDAC, mTOR, CDK, Aurora Kinase, JAK, etc., in lung cancer, breast cancer, leukemia, lymphoma, etc.
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

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Apoptosis
Autophagy
Endogenous Metabolite
5-HT Receptor
Antibacterial
Adrenergic Receptor
DNA/RNA Synthesis
Dopamine Receptor
Antibiotic
VEGFR
COX
Potassium Channel
Calcium Channel
Histamine Receptor
Sodium Channel
EGFR
Parasite
PI3K
ROS
Cytochromes P450
CDK
Reactive Oxygen Species
FLT
NF-κB
JAK
PDGFR
Glucocorticoid Receptor
HIV Protease
FGFR
c-Kit
Topoisomerase
mTOR
HDAC
Akt
Microtubule Associated
c-Met/HGFR
PPAR
Virus Protease
Ferroptosis
AChR
Prostaglandin Receptor
SARS-CoV
Src
Dehydrogenase
Nucleoside Antimetabolite/Analog
GABA Receptor
p38 MAPK
Estrogen Receptor/ERR
Antifungal
Mitophagy
iGluR
ERK
Interleukin
Estrogen/progestogen Receptor
Bcr-Abl
Tyrosine Kinases
Adenosine Receptor
Influenza Virus
Caspase
Androgen Receptor
Ras
Raf
GPCR
TNF
Epigenetic Reader Domain
PARP
HSV
HSP
Aurora Kinase
P-gp
PDE
Bcl-2 Family
Serotonin Transporter
TRP/TRPV Channel
MEK
ALK
MDM-2/p53
HBV
HER
Trk receptor
HIF/HIF Prolyl-Hydroxylase
Histone Methyltransferase
PKC
STAT
Opioid Receptor
Mitochondrial Metabolism
RAAS
c-RET
Norepinephrine
TLR
ATPase
c-Fms
HCV Protease
Phosphatase
NMDAR
ROS Kinase
Endothelin Receptor
AMPK
Beta Amyloid
DNA Alkylator/Crosslinker
Wnt/beta-catenin
JNK
Drug Metabolite
FAK
E1/E2/E3 Enzyme
MMP
Chk
GSK-3
TAM Receptor
LPL Receptor
Molecular Glues
Proton pump
Retinoid Receptor
Gamma-secretase
S1P Receptor
Progesterone Receptor
Kras
SGLT
Guanylate cyclase
CXCR
NO Synthase
GluR
IGF-1R
CFTR
Reverse Transcriptase
TGF-beta/Smad
Antifolate
Nrf2
p53
Carbonic Anhydrase
IL Receptor
HIF
DNA-PK
P2X Receptor
ROCK
S6 Kinase
Antioxidant
Syk
Vasopressin Receptor
Proteasome
PKA
DNA Alkylation
ATM/ATR
HMG-CoA Reductase
Transferase
ADC Cytotoxin
IAP
PLK
GNRH Receptor
Hedgehog/Smoothened
Ligands for E3 Ligase
Indoleamine 2,3-Dioxygenase (IDO)
Kinesin
IDO
Anti-infection
Monoamine Oxidase
P2Y Receptor
Angiotensin-converting Enzyme (ACE)
MAPK
MAO
Isocitrate Dehydrogenase (IDH)
Lipoxygenase
DHFR
Integrin
CSF-1R
BTK
MRP
RIP kinase
Antifection
OX Receptor
DNA Methyltransferase
Glutathione Peroxidase
Leukotriene Receptor
Cannabinoid Receptor
Histone Demethylase
Sirtuin
Casein Kinase
Serine Protease
Mdm2
PAK
IRAK
IκB/IKK
Antiviral
DNA
Hydroxylase
Sigma receptor
Smo
Phospholipase
Neurokinin receptor
Pim
FXR
Bradykinin Receptor
PROTACs
CCR
Glucagon Receptor
Ephrin Receptor
PD-1/PD-L1
Reductase
Tie-2
IKZF
PYK2
IFNAR
Telomerase
Thrombin
NOD-like Receptor (NLR)
Serine/threonin kinase
Xanthine Oxidase
STING
Tyrosinase
PERK
Cholinesterase (ChE)
DPP-4
GPCR19
RSV
CRFR
GHSR
NOD
CRM1
Glutaminase
Fatty Acid Synthase
Somatostatin
Wee1
PGE Synthase
YAP
NADPH
Na-K-Cl cotransporter
Neuropeptide Y Receptor
CaMK
AhR
Chloride channel
Melatonin Receptor
Aryl Hydrocarbon Receptor
CGRP Receptor
ABC Transporter
Monoamine Transporter
glycosidase
DUB
c-Myc
CaSR
Photosensitizer
NAMPT
GST
Aromatase
Oxytocin Receptor
Cholecystokinin Receptor
Glucosidase
BCRP
Survivin
Aminopeptidase
Cuproptosis
Discoidin Domain Receptor (DDR)
Protease-activated Receptor
Annexin A
MT Receptor
transporter
IRE1
KSP
OXPHOS
Free radical scavengers
FKBP
MLK
LTR
ATP Citrate Lyase
ribosome
ROR
OAT
Rho
Melanocortin Receptor
Gap Junction Protein
Beta-Secretase
Decarboxylase
Adenosine Deaminase
UGT
Thrombopoietin Receptor
p97
Necroptosis
RANKL/RANK
GRK
LPA Receptor
PDK
SGK
NOS
Monocarboxylate transporter
Cysteine Protease
LDL
DNA gyrase
NEDD8
VDA
PROTAC Linker
Porcupine
CD73
Amino Acids and Derivatives
Ligands for Target Protein for PROTAC
Galectin
Hexokinase
PI4K
Complement System
Arginase
DYRK
HCN Channel
Histone Acetyltransferase
PAI-1
TOPK
Acyltransferase
MIF
Neurotensin Receptor
Adenylate cyclase
GlyT
ASK
Methionine Adenosyltransferase (MAT)
Aquaporin
Advanced Glycation End Products
Cell wall
OCT
Hck
Stemness kinase
ACK1
Lipid
PSMA
BMI-1
RAR/RXR
MALT
MyD88
Cadherin
Huntingtin
GluCls
Pyroptosis
RXFP receptor
NADPH-oxidase
Hydrogenase
Factor VIIa
N-Acetylglucosaminyltransferase
ATG
Anion Exchanger
E3 Ligase Ligand-Linker Conjugates
Hippo pathway
Imidazoline Receptor
MicroRNA
Cell Cycle Arrest
LIM Kinase
Glucokinase
PAFR
MTH1
HCAR
MNK
KLF
GTPase
Factor Xa
Liver X Receptor
MELK
Thyroid hormone receptor(THR)
NPC1L1
Kisspeptin
Myosin
Thioredoxin
Neprilysin
FOXO
Liposome
Vitamin
Drug-Linker Conjugates for ADC
Ferroportin
PGC-1α

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