Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Auglurant is a novel and selective mGlu5 antagonist (IC50: 11 nM (rat) and an IC50: 14 nM (human)). Auglurant has an acceptable CNS penetration.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
5 mg | 6-8 weeks | $ 446.00 | |
25 mg | 6-8 weeks | $ 1,430.00 | |
50 mg | 6-8 weeks | $ 1,860.00 | |
100 mg | 6-8 weeks | $ 2,500.00 | |
1 mL * 10 mM (in DMSO) | 6-8 weeks | $ 432.00 |
Description | Auglurant is a novel and selective mGlu5 antagonist (IC50: 11 nM (rat) and an IC50: 14 nM (human)). Auglurant has an acceptable CNS penetration. |
Targets&IC50 | mGluR5 (rat):11 nM (IC50), mGluR5 (human):14 nM (IC50) |
Synonyms | VU0424238 |
Molecular Weight | 325.3 |
Formula | C16H12FN5O2 |
CAS No. | 1396337-04-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
You can also refer to dose conversion for different animals. More
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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
Auglurant 1396337-04-4 Others VU0424238 VU 0424238 VU-0424238 inhibitor inhibit