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AR-9281

Catalog No. T14315   CAS 913548-29-5
Synonyms: APAU

AR-9281 (APAU) is a potent and selective inhibitor of soluble epoxide hydrolase (s-EH) potentially for the treatment of hypertension and type 2 diabetes

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
AR-9281 Chemical Structure
AR-9281, CAS 913548-29-5
Pack Size Availability Price/USD Quantity
1 mg In stock $ 57.00
2 mg In stock $ 81.00
5 mg In stock $ 117.00
10 mg In stock $ 176.00
25 mg In stock $ 316.00
50 mg In stock $ 475.00
100 mg In stock $ 695.00
1 mL * 10 mM (in DMSO) In stock $ 137.00
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Biological Description
Chemical Properties
Storage & Solubility Information
Description AR-9281 (APAU) is a potent and selective inhibitor of soluble epoxide hydrolase (s-EH) potentially for the treatment of hypertension and type 2 diabetes
Synonyms APAU
Molecular Weight 319.44
Formula C18H29N3O2
CAS No. 913548-29-5

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

Solubility Information

DMSO: 25 mg/mL (78.26 mM), sonification is recommended.

TargetMolReferences and Literature

1. Chen D, et al. Pharmacokinetics and pharmacodynamics of AR9281, an inhibitor of soluble epoxide hydrolase, in single- and multiple-dose studies in healthy human subjects. J Clin Pharmacol. 2012 Mar;52(3):319-28.

Related compound libraries

This product is contained In the following compound libraries:
Bioactive Compounds Library Max Bioactive Compound Library Anti-Hypertension Compound Library Inhibitor Library NO PAINS Compound Library Anti-Aging Compound Library Anti-Diabetic Compound Library ReFRAME Related Library Metabolism Compound Library Anti-Metabolism Disease Compound Library

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CUDA (Rac)-EC5026 Dual FAAH/sEH-IN-1 VU534 beta-Amyrin acetate Diflapolin PTUPB BI-1935

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

AR-9281 913548-29-5 Metabolism Epoxide Hydrolase inflammation hypertension AR9281 APAU MsEH HsEH soluble epoxide hydrolase (s-EH) oral inhibit Inhibitor AR 9281 type 2 diabetes inhibitor

 

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