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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10240 | ACP-5862 | BTK | |
ACP-5862 is a major active and pyrrolidine ring-opened metabolite of Acalabrutinib (IC50: 5.0 nM for BTK). Acalabrutinib is an irreversible and highly selective BTK inhibitor (IC50: 3 nM; EC50: 8 nM). |