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Home > Cytoskeletal Signaling > Akt > A-674563

A-674563

Catalog No. T6139    CAS 552325-73-2    Synonyms: A674563, A 674563,

A-674563 is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC.

Pack Size Availability Price/USD Quantity
1 mg Inquiry 67.00
2 mg Inquiry 120.00
5 mg Inquiry 160.00
10 mg Inquiry 260.00
25 mg Inquiry 585.00
50 mg Inquiry 780.00
1 mL * 10 mM (in DMSO) Inquiry 160.00
Bulk Size: Please Quote for Discount Please Quote for Bulk Size
Biological Activity:

Product Description:

A-674563 is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC.

Receptor:

Akt1; CDK2; ERK2; GSK-3β; PKA;

Chemical Information:
Molecular Weight 358.44
Formula C22H22N4O
CAS Number 552325-73-2
Solubility

DMSO: 67 mg/mL (186.9 mM)

Ethanol: 15 mg/mL (41.8 mM)

Water: 66 mg/mL (184.1 mM)

( < 1 mg/ml refers to the product slightly soluble or insoluble )
Storage store at -80°C
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.