Powder: -20°C for 3 years | In solvent: -80°C for 1 year
(±)-Anatoxin A fumarate is a natural alkaloid isolated from freshwater cyanobacterium. It is a potent nicotinic receptor agonist and exhibits Ki values of 1.25 nM and 1.84 μM for binding to putative α4β2-type nAChR and α7-type nAChR in rat brain membranes, respectively. (±)-Anatoxin A fumarate stimulates [3H]-dopamine release from rat striatal synaptosomes with EC50 of 134 nM.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | 35 days | $ 597.00 |
Description | (±)-Anatoxin A fumarate is a natural alkaloid isolated from freshwater cyanobacterium. It is a potent nicotinic receptor agonist and exhibits Ki values of 1.25 nM and 1.84 μM for binding to putative α4β2-type nAChR and α7-type nAChR in rat brain membranes, respectively. (±)-Anatoxin A fumarate stimulates [3H]-dopamine release from rat striatal synaptosomes with EC50 of 134 nM. |
Targets&IC50 | α7 receptor:1.84 μM (Ki), α4β2 receptor:1.25 nM (Ki) |
Molecular Weight | 281.3 |
Formula | C14H19NO5 |
CAS No. | 1219922-30-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
H2O: Soluble
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(±)-Anatoxin A fumarate 1219922-30-1 Others (±) Anatoxin A fumarate Anatoxin A Fumarate (±)Anatoxin A fumarate inhibitor inhibit