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Compound Libraries Kinase Inhibitor Library

Kinase Inhibitor Library

Catalog No. L1600
  Library Compound List   Excel SDF

In biochemistry, a kinase is an enzyme that catalyzes the transfer of phosphate groups from high-energy, phosphate-donating molecules (ATP) to specific substrates. This process is known as phosphorylation. The protein kinases make up the majority of all kinases and are widely studied. A protein kinase modifies other molecules, mostly proteins, by phosphorylation to regulate the majority of cellular pathways, especially those involved in signal transduction. Various other kinases act on small molecules such as lipids, carbohydrates, amino acids, and nucleotides, either for signaling or to prime them for metabolic pathways.

TargetMol’s Tyrosine Kinase Inhibitors Library, containing 2203 kinase inhibitors, can be used for research in chemical genomics, pharmacological study, and drug screening for related diseases.

Pack Size Price/USD
100 μL * 10 mM (in DMSO) 28522.00
250 μL * 10 mM (in DMSO) 46734.00
1 mg 46734.00
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Product Description

  • A unique collection of 2203 kinase inhibitors for high throughput screening and high content screening for drug discovery in kinase related diseases;
  • Bioactivity and safety confirmed by pre-clinical research and clinical trials, and some of them are approved by FDA;
  • Targets include MAPK, PI3K, JAK, STAT, CDK, MEK, Insulin/IGF receptors, CaM Kinease II, PKA, JNK, PKC, RAF, EGFR, SAPK, GSK, MLCK, Src-family, IKK, PDGFR, VEGFR, etc;
  • Detailed compound information with structure, target, activity, IC50 value, and biological activity description;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality;

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L1600)

Library Composition

ERK (152)
PI3K (120)
VEGFR (111)
CDK (110)
EGFR (102)
PKM (84)
Src (69)
mTOR (67)
FLT (66)
Glucokinase (63)
JAK (63)
PLK (62)
PDGFR (59)
FGFR (57)
ATM/ATR (56)
c-Kit (52)
PKC (51)
Raf (51)
Bcr-Abl (50)
MAPK (50)
p38 MAPK (48)
c-Met/HGFR (47)
Akt (45)
GSK-3 (43)
ALK (42)
JNK (37)
Tyrosine Kinases (37)
AMPK (36)
Streptokinase (34)
MEK (32)
DNA-PK (31)
DYRK (29)
Aurora Kinase (29)
IκB/IKK (27)
BTK (26)
NF-κB (26)
TAM Receptor (24)
Casein Kinase (24)
c-RET (23)
HER (23)
S6 Kinase (23)
TNF (22)
Trk receptor (22)
ROCK (21)
ROS (21)
Streptokinase A (21)
PKA (21)
CaMK (21)
Autophagy (19)
STAT (18)
Ras (17)
LRRK2 (17)
IGF-1R (16)
Chk (16)
Tyrosinase (16)
Syk (16)
TGF-beta/Smad (15)
Pim (15)
FAK (15)
Serine/threonin kinase (14)
AChR (13)
Apoptosis (12)
Potassium Channel (12)
S1P Receptor (10)
PDK (10)
5-HT Receptor (10)
Antiviral (10)
CSF-1R (10)
c-Fms (10)
Adrenergic Receptor (9)
IL Receptor (9)
Serine Protease (9)
PPAR (8)
PERK (8)
Phosphoglycerate kinase, glycosomal (8)
DNA/RNA Synthesis (8)
Ephrin Receptor (7)
Epigenetic Reader Domain (7)
COX (7)
Caspase (7)
LIM Kinase (7)
P450 (7)
Plasmodium falciparum (7)
Rho (6)
Sodium Channel (6)
SGK (6)
PAK (6)
Tie-2 (6)
GRK (6)
Endogenous Metabolite (6)
Antioxidant (6)
ATPase (6)
Beta-lactamase AmpC (5)
Ataxin (5)
Discoidin Domain Receptor (DDR) (5)
Dehydrogenase (5)
Hexokinase (5)
Histamine Receptor (5)
HSP (5)
MLK (5)
PDE (5)
NADPH (4)
PYK2 (4)
Topoisomerase (4)
Wnt/beta-catenin (4)
MNK (4)
Mothers against decapentaplegic homolog 3 (4)
IRE1 (4)
Carbonic Anhydrase (4)
Dopamine Receptor (4)
E1/E2/E3 Enzyme (4)
Estrogen/progestogen Receptor (4)
BCL (4)
Calcium Channel (3)
ASK (3)
ACK (3)
Adenosine Receptor (3)
Antibacterial (3)
Antibiotic (3)
DNA Alkylation (3)
c-Myc (3)
Integrin (3)
Interleukin Related (3)
Kinesin (3)
Mitochondrial Metabolism (3)
Lipoxygenase (3)
Microtubule Associated (3)
Histone Methyltransferase (3)
HIV Protease (3)
Hck (3)
HDAC (3)
GluR (3)
Geminin (3)
Vitamin (3)
PTEN (3)
Prelamin-A/C (3)
Prostaglandin Receptor (3)
Na-K-Cl cotransporter (3)
NAMPT (2)
OXPHOS (2)
Nrf2 (2)
Nuclear factor erythroid 2-related factor 2 (2)
Nonstructural protein 1 (2)
NOS (2)
Phosphatase (2)
Parasite (2)
PARP (2)
Phospholipase (2)
Phosphorylase (2)
PI4K (2)
PGK (2)
Proteasome (2)
RIP kinase (2)
ROR (2)
SIK (2)
Sirtuin (2)
Wee1 (2)
Wnk (2)
TOPK (2)
GABA Receptor (2)
HIF (2)
HSV (2)
Guanine nucleotide-binding protein G(s), subunit alpha (2)
HEK293 (2)
Microtubule-associated protein tau (2)
MELK (2)
microRNA 21 (2)
MAO (2)
Mitophagy (2)
MMP (2)
MPO (2)
KSP (2)
LDL (2)
Chloride channel (2)
cholecystokinin (2)
Cysteine Protease (2)
Antifection (2)
Apoptosis inducer (2)
Aromatase (2)
AhR (2)
Beta Amyloid (2)
ATP Citrate Lyase (2)
BACE (2)
Autoinducer 1 sensor kinase/phosphatase luxN (1)
ATPase family AAA domain-containing protein 5 (1)
BMI-1 (1)
APC (1)
advanced glycation end products (1)
DNA Alkylator/Crosslinker (1)
DNA (1)
FAAH (1)
cell cycle arrest (1)
DHFR (1)
CXCR (1)
Leukotriene Receptor (1)
Lipid (1)
lysosomal autophagy (1)
IRAK (1)
Immunology & Inflammation related (1)
Inositol monophosphatase 1 (1)
Monoamine Transporter (1)
Melatonin Receptor (1)
Histone Demethylase (1)
Hippo pathway (1)
Hedgehog/Smoothened (1)
HCV Protease (1)
Gap Junction Protein (1)
Glucagon Receptor (1)
Glucagon-like peptide 1 receptor (1)
Fatty Acid Synthase (1)
Ferroptosis (1)
Free radical scavengers (1)
Glycoprotein hormones alpha chain (1)
GPR (1)
GPX (1)
GST (1)
GTPase (1)
TLR (1)
Thrombin (1)
TAR DNA-binding protein 43 (1)
Transferase (1)
transporter (1)
Stemness kinase (1)
Survival motor neuron protein (1)
Sigma receptor (1)
Salt-Inducible Kinase (1)
RAAS (1)
Proton pump (1)
P-gp (1)
p53 (1)
PAI-1 (1)
NPC1L1 (1)
Norepinephrine (1)
P2 Receptor (1)
Neurokinin receptor (1)
NOD-like Receptor (NLR) (1)
Myosin (1)