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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T10823 | Trans-Pralsetinib | cis-Pralsetinib,cis-BLU-667 | c-RET |
trans-Pralsetinib (trans-BLU-667) is an inhibitor of rearranged during transfection (RET). | |||
TQ0277L | Pralsetinib HCl (2097132-94-8 free base) | Pralsetinib HCl,Pralsetinib hydrochloride,BLU-667,BLU667,BLU 667 | |
Pralsetinib is a selective and next-generation RET inhibitor (IC50: 0.3-0.4 nM for WT RET, RET mutants V804L, V804M, M918T, and CCDC6-RET fusion). BLU-667 is an effective and selective inhibitor of RET mutations, fusions... | |||
TQ0277 | Pralsetinib | Blu667 | c-RET |
Pralsetinib (Blu667) (BLU-667) is a highly potent, selective RET inhibitor (IC50s: 0.4, 0.3, 0.4, 0.4, and 0.4 nM for WT RET, RET mutants V804L, V804M, M918T and CCDC6-RET fusion). |