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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T33945 | PF-06260933 HCl | PF06260933 dihydrochloride,PF-06260933 dihydrochloride,PF 06260933 dihydrochloride | Others |
PF-06260933 Dihydrochloride is a MAP4K4 (HGK) inhibitor (IC50 = 140 nM). It can improve the fasting hyperglycemia in mice. In addition, it inhibited Mink and Tnik (IC50 values of 8 and 13 nM, respectively). | |||
T36016 | PF 06260933 dihydrochloride | Others | |
MAP4K4 (HGK) inhibitor (IC50 = 140 nM). Also inhibits MINK and TNIK (IC50 values are 8 and 13 nM, respectively). Improves fasting hyperglycemia in mice. Orally active. Ammirati et al (2015) Discovery of an in vivo tool t... |