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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T12183 | Nav1.7-IN-3 | Others | |
Nav1.7-IN-3 is a selective and orally bioavailable inhibitor of voltage-gated sodium channel Nav1.7(IC50 of 8 nM). | |||
T37093 | 4,9-Anhydrotetrodotoxin | 4,9-Anhydrotetrodotoxin,4,9-anhydro-TTX | |
4,9-Anhydrotetrodotoxin (4,9-anhydro-TTX) is a derivative of TTX that selectively blocks inward sodium current through Nav1.6 voltage-activated sodium channels (IC50 = 7.8 nM in Xenopus oocytes). [1][2][3] It demonstrate... | |||
TP1972 | OD1 | ||
Potent rat Nav1.7, human Nav1.4 and rat Nav1.6 channel activator (EC50 values are 7, 10 and 47 nM, respectively). Exhibits minimal activation at mammalian Nav1.2, Nav1.3 and Nav1.5 (EC50 values >3 μM). Inhibits fast inac... |