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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T39410 | Zevaquenabant | (S)-MRI-1867 | |
Zevaquenabant ((S)-MRI-1867), a dual cannabinoid CB1 receptor and inducible NOS (iNOS) antagonist, is orally bioavailable and peripherally restricted. It effectively mitigates obesity-induced chronic kidney disease (CKD)... | |||
T39074 | (Rac)-Zevaquenabant | (Rac)-MRI-1867,(Rac)-Zevaquenabant | |
(Rac)-Zevaquenabant ((Rac)-MRI-1867, compound 6b) is a potent and selective antagonist of the cannabinoid receptor type 1 (CB1R) and inducible nitric oxide synthase (iNOS), exhibiting a binding affinity (Ki) of 5.7 nM sp... |