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Home > Cell cycle/Check point > PAK > PF-3758309
PF-3758309  
Catalog No. T6626    CAS 898044-15-0
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Availability
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5mg
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54.00
10mg
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78.00
25mg
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140.00
50mg
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253.00
100mg
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429.00
200mg
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772.00
1 mL * 10 mM (in DMSO)
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59.00
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Documents and Quality Management
Purity:98.00% COA Datasheet
Biological Activity:

Product Description:

PF-03758309 (IC50=1.3 nM), a pyrrolopyrazole inhibitor of PAK4, has effective ATP-competition.

Target:
PAK5; PAK6; PAK1; PAK4; PAK5 ; PAK6 ; PAK1 ; PAK4;
Research Area:
cancer
Chemical Information:
Molecular Weight 490.62
Formula C25H30N8OS
CAS Number 898044-15-0
Solubility DMSO:91 mg/mL (185.5 mM);Ethanol:91 mg/mL (185.5 mM);Water:<1 mg/mL
Storage 3 years -20°C powder;
2 years -80°C in solvent;
Remark For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20 ℃ for several month.
Technical Support

Answers to questions you may have can be found in the inhibitor handling instructions. Topics include how to prepare stock solutions, how to store Products, and issues that need special attention for cell-based assays and animal experiments.

Related Compound Libraries
This product is contained In the following compound libraries:
  • The compound is not included in our libraries at this moment.
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Reference

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