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Histrelin acetate

🥰Excellent
Catalog No. TP2107LCas No. 220810-26-4
Alias Histrelin acetate(76712-82-8 free base)

Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It acts on particular cells of the pituitary gland called gonadotropes when present in the bloodstream. Histrelin stimulates these cells to release luteinizing hormone and follicle-stimulating hormone. Thus it is considered a gonadotropin-releasing hormone agonist or GnRH agonist.

Histrelin acetate
Other Forms of Histrelin acetate:
HistrelinT2130876712-82-8
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Histrelin acetate

🥰Excellent
Purity: 99.92%
Catalog No. TP2107LAlias Histrelin acetate(76712-82-8 free base)Cas No. 220810-26-4
Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It acts on particular cells of the pituitary gland called gonadotropes when present in the bloodstream. Histrelin stimulates these cells to release luteinizing hormone and follicle-stimulating hormone. Thus it is considered a gonadotropin-releasing hormone agonist or GnRH agonist.
Pack SizePriceUSA WarehouseGlobal WarehouseQuantity
1 mg$80In StockIn Stock
5 mg$178In StockIn Stock
10 mg$289In StockIn Stock
25 mg$489In StockIn Stock
50 mg$686In StockIn Stock
100 mg$969In StockIn Stock
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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]
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Purity:99.92%
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COA HPLC MS

Product Introduction

Bioactivity
Description
Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency. It acts on particular cells of the pituitary gland called gonadotropes when present in the bloodstream. Histrelin stimulates these cells to release luteinizing hormone and follicle-stimulating hormone. Thus it is considered a gonadotropin-releasing hormone agonist or GnRH agonist.
SynonymsHistrelin acetate(76712-82-8 free base)
Chemical Properties
Molecular Weight1383.55
FormulaC68H90N18O14
Cas No.220810-26-4
SmilesCCNC([C@@H]1CCCN1C([C@H](CCCNC(N)=N)NC([C@H](CC(C)C)NC([C@@H](CC2=CN(C=N2)CC3=CC=CC=C3)NC([C@H](CC4=CC=C(C=C4)O)NC([C@H](CO)NC([C@H](CC5=CNC6=CC=CC=C65)NC([C@H](CC7=CNC=N7)NC([C@@H]8CCC(N8)=O)=O)=O)=O)=O)=O)=O)=O)=O)=O.CC(O)=O
Relative Density.no data available
Sequence{Pyr}-His-Trp-Ser-Tyr-{d-His(Bzl)}-Leu-Arg-Pro-{NHEt}
Sequence Short{Pyr}-HWSY-{d-His(Bzl)}-LRP-{NHEt}
Storage & Solubility Information
Storagekeep away from moisture | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.
Solubility Information
DMSO: Soluble

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TargetMol | Animal experimentsFor example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。
Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSOTargetMol | reagent (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
Preparation method for in vivo formula: Take 50 μL DMSOTargetMol | reagent main solution, add 300 μLPEG300TargetMol | reagent mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2OTargetMol | reagent mix well and clarify
For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.
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Keywords

Histrelin acetateHistrelin AcetateGNRHReceptorGNRHRGNRH Receptor
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