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CB2R/FAAH modulator-1
🥰Excellent
Catalog No. T67896Cas No. 928892-60-8
CB2R/FAAH modulator-1, a cannabinoid type 2 receptor (CB2R) agonist, is also a fatty acid amide hydrolase (FAAH) inhibitor (IC50=4 μM) that reduces the production of pro-inflammatory and anti-inflammatory cytokines and is commonly used in inflammation studies. The Kis for CB2R and CB1R are 14.8 nM and 241.3 nM, respectively.
CB2R/FAAH modulator-1
🥰Excellent
Purity: 99.77%
Catalog No. T67896Cas No. 928892-60-8
CB2R/FAAH modulator-1, a cannabinoid type 2 receptor (CB2R) agonist, is also a fatty acid amide hydrolase (FAAH) inhibitor (IC50=4 μM) that reduces the production of pro-inflammatory and anti-inflammatory cytokines and is commonly used in inflammation studies. The Kis for CB2R and CB1R are 14.8 nM and 241.3 nM, respectively.
| Pack Size | Price | Availability | Quantity |
|---|---|---|---|
| 1 mg | $48 | In Stock | |
| 5 mg | $113 | In Stock | |
| 10 mg | $165 | In Stock | |
| 25 mg | $248 | In Stock | |
| 50 mg | $348 | In Stock | |
| 100 mg | $475 | In Stock | |
| 200 mg | $639 | In Stock | |
| 1 mL x 10 mM (in DMSO) | $116 | In Stock |
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Purity:99.77%
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Product Introduction
Bioactivity
Chemical Properties
| Description | CB2R/FAAH modulator-1, a cannabinoid type 2 receptor (CB2R) agonist, is also a fatty acid amide hydrolase (FAAH) inhibitor (IC50=4 μM) that reduces the production of pro-inflammatory and anti-inflammatory cytokines and is commonly used in inflammation studies. The Kis for CB2R and CB1R are 14.8 nM and 241.3 nM, respectively. |
| Targets&IC50 | CB2 receptor:14.8 nM (Kis), CB1 receptor:489 nM (EC50), CB2 receptor:123.6 nM (EC50), CB1 receptor:241.3 nM (Kis), FAAH:4 μM |
| In vitro | CB2R/FAAH modulator-1 (compound 13; 10 μM; 24 h) reduces TNFα, IFN-γ, IL-1β, and IL-6 production in unstimulated monocytes and macrophages[1]. |
| Molecular Weight | 361.48 |
| Formula | C24H27NO2 |
| Cas No. | 928892-60-8 |
| Smiles | N(C(=O)C1=C(OCC2=CC=CC=C2)C=CC=C1)C34CC5CC(C3)CC(C4)C5 |
| Relative Density. | 1.19 g/cm3 (Predicted) |
Storage & Solubility Information
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||
| Solubility Information | DMSO: 11 mg/mL (30.43 mM), Sonication is recommended.  | |||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||
DMSO
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In Vivo Formulation Calculator (Clear solution)
Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:
For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . A total of 10 animals were administered, and the formula you used is 5% 
DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH2O. So your working solution concentration is 2 mg/mL。Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO (mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.
(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.Preparation method for in vivo formula: Take 50 μL DMSO main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarify
main solution, add 300 μLPEG300 mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH2O mix well and clarifyFor Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.
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