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WH-4-025

Catalog No. T9219 CAS 1876463-35-2

WH-4-025 is a Salt-inducible kinase (SIK) inhibitor.

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WH-4-025, CAS 1876463-35-2

Pack Size	Availability	Price/USD
2 mg	In stock	59.00
5 mg	In stock	85.00
10 mg	In stock	142.00
25 mg	In stock	279.00
50 mg	In stock	441.00
100 mg	In stock	693.00
200 mg	In stock	1039.00

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Purity 98.70%

HNMR HPLC COA

Datasheet

Biological Description

Chemical Properties

Storage & Solubility Information

Description

WH-4-025 is a Salt-inducible kinase (SIK) inhibitor.

Molecular Weight	741.76
Formula	C39H38F3N7O5
CAS No.	1876463-35-2

Storage

Powder: -20°C for 3 years

In solvent: -80°C for 6 months

Solubility Information

DMSO: 125 mg/mL (164.47 mM, Need ultrasonic

( < 1 mg/ml refers to the product slightly soluble or insoluble )

Citations

References and Literature

1. Brookline Avenue, et al. USES OF SALT-INDUCIBLE KINASE (SIK) INHIBITORS. Patent WO2016023014A2.

Related Products

Related compounds with same targets

WH-4-025 ARN-3236 YKL-06-061 YKL-05-099

Dose Conversion

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Calculation results:

Working concentration: mg/ml;

Method for preparing DMSO master liquid: mg drug pre-dissolved in μL DMSO (Master liquid concentration mg/mL)，Please contact us first if the concentration exceeds the DMSO solubility of the batch of drug.

Method for preparing in vivo formulation：Take μL DMSO master liquid, next add μL PEG300， mix and clarify, next add μL Tween 80，mix and clarify, next add μL ddH₂O, mix and clarify.

Note:

Be sure to add the solvent(s) in order. Physical methods such as vortex, ultrasound or hot water bath can be used to aid dissolving.

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What is the mass of compound required to make a 10 mM stock solution in 10 ml of water given that the molecular weight of the compound is 197.13 g/mol?
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The answer of 19.713 mg appears in the Mass box

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What volume of a given 10 mM stock solution is required to make 20ml of a 50 μM solution?
Using the equation C1V1 = C2V2, where C1=10 mM, C2=50 μM, V2=20 ml and V1 is the unknown:
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The answer of 100 microliter (0.1 ml) appears in the Volume (start) box

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Molar mass (molar weight) is the mass of one mole of a substance and is expressed in g/mol.

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Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.