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SR-3029

Name: SR-3029
Brand: TargetMol
SKU: T3972
Price: 30 USD
Availability: InStock
Rating: 5 (10 reviews)

🥰Excellent

Catalog No. T3972Cas No. 1454585-06-8

Alias SR3029

SR-3029 is a highly potent and specific inhibitor of CK1δ/CK1ε.

SR-3029

🥰Excellent

Purity: 99.64%

Catalog No. T3972Alias SR3029Cas No. 1454585-06-8

SR-3029 is a highly potent and specific inhibitor of CK1δ/CK1ε.

Pack Size	Price	Availability
1 mg	$30	In Stock
5 mg	$73	In Stock
10 mg	$119	In Stock
25 mg	$257	In Stock
50 mg	$413	In Stock
1 mL x 10 mM (in DMSO)	$77	In Stock

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Batch Information

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Purity:99.64%

Resource Download

COA LCMS HNMR

Product Introduction

Bioactivity

Description	SR-3029 is a highly potent and specific inhibitor of CK1δ/CK1ε.
Targets&IC50	Cdk4-CyclinD1:576 nM, CDK6-CyclinD1:428 nM, FLT3:3000 nM, CK1δ:44 nM, CK1ε:260 nM, CDK4-CyclinD3:368 nM, CDK6-CyclinD3:427 nM
Synonyms	SR3029

Chemical Properties

Molecular Weight	480.45
Formula	C₂₃H₁₉F₃N₈O
Cas No.	1454585-06-8
Smiles	Fc1cccc(c1)-n1cnc2c(NCc3nc4ccc(F)c(F)c4[nH]3)nc(nc12)N1CCOCC1
Relative Density.	1.62 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 45 mg/mL (93.66 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	2.0814 mL	10.4069 mL	20.8138 mL	104.0691 mL
5 mM	0.4163 mL	2.0814 mL	4.1628 mL	20.8138 mL
10 mM	0.2081 mL	1.0407 mL	2.0814 mL	10.4069 mL
20 mM	0.1041 mL	0.5203 mL	1.0407 mL	5.2035 mL
50 mM	0.0416 mL	0.2081 mL	0.4163 mL	2.0814 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the mother liquor preparation method and in vivo formula preparation method:

For example, your dosage is 10 mg/kg Each animal weighs 20 g, and the dosage volume is 100 μL . TargetMol | Animal experiments

A total of 10 animals were administered, and the formula you used is 5% TargetMol | reagent

DMSO+30% PEG300+5% Tween 80+60% Saline/PBS/ddH₂O. So your working solution concentration is 2 mg/mL。

Mother liquor preparation method: 2 mg of drug dissolved in 50 μL DMSO TargetMol | reagent

(mother liquor concentration of 40 mg/mL), if you need to configure a concentration that exceeds the solubility of the product, please contact us first.

Preparation method for in vivo formula: Take 50 μL DMSO TargetMol | reagent

main solution, add 300 μLPEG300 TargetMol | reagent

mix well and clarify, then add 50 more μL Tween 80, mix well and clarify, then add 600 more μLSaline/PBS/ddH₂O TargetMol | reagent

mix well and clarify

For Reference Only. Please develop an appropriate dissolution method based on your laboratory animals and route of administration.

All types of co-solvents required for the protocol, such asDMSO, PEG300/ PEG400, Tween 80, SBE-β-CD, corn oil are available for purchase on the TargetMol website with a simple click.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Sci Citations

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc