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Protein kinase inhibitor peptide

Catalog No. TP2349 CAS 128022-93-5

Synonyms: PKIP

Protein kinase inhibitor peptide matches the inhibitory domain of the heat-stable protein kinase inhibitor.

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Protein kinase inhibitor peptide Chemical Structure

Protein kinase inhibitor peptide, CAS 128022-93-5

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Biological Description

Chemical Properties

Storage & Solubility Information

Description

Protein kinase inhibitor peptide matches the inhibitory domain of the heat-stable protein kinase inhibitor.

Synonyms	PKIP
Molecular Weight	1970.15
Formula	C84H136N28O27
CAS No.	128022-93-5

Storage

keep away from moisture

Powder: -20°C for 3 years | In solvent: -80°C for 1 year

References and Literature

1. Dalton GD, Dewey WL. Protein kinase inhibitor peptide (PKI): a family of endogenous neuropeptides that modulate neuronal cAMP-dependent protein kinase function. Neuropeptides. 2006 Feb;40(1):23-34. Epub 2006 Jan 26. Review. PubMed PMID: 16442618. 2. Olah GA, Mitchell RD, Sosnick TR, Walsh DA, Trewhella J. Solution structure of the cAMP-dependent protein kinase catalytic subunit and its contraction upon binding the protein kinase inhibitor peptide. Biochemistry. 1993 Apr 13;32(14):3649-57. PubMed PMID: 8385485. 3. Taffs RE, Sitkovsky MV. Modulation of the effector functions of cytolytic T-lymphocytes with synthetic peptide inhibitors of protein kinases. J Pharm Sci. 1992 Jan;81(1):37-44. PubMed PMID: 1619567. 4. Glass DB, Feller MJ, Levin LR, Walsh DA. Structural basis for the low affinities of yeast cAMP-dependent and mammalian cGMP-dependent protein kinases for protein kinase inhibitor peptides. Biochemistry. 1992 Feb 18;31(6):1728-34. PubMed PMID: 1310617.

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Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.

Keywords

Protein kinase inhibitor peptide 128022-93-5 PKIP inhibitor inhibit

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