Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PROTAC Sirt2 Degrader-1 is a SirReal-based PROTAC, acts as a Sirt2 degrader, composed of a highly potent and isotype-selective Sirt2 inhibitor, a linker, and a bona fide cereblon ligand for E3 ubiquitin ligase. PROTAC Sirt2 Degrader-1 shows an IC50 of 0.25 μM for Sirt2, with no effect on Sirt1/Sirt3 (IC50s < 100 μM)[1].
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500 mg | Inquiry | Inquiry |
Description | PROTAC Sirt2 Degrader-1 is a SirReal-based PROTAC, acts as a Sirt2 degrader, composed of a highly potent and isotype-selective Sirt2 inhibitor, a linker, and a bona fide cereblon ligand for E3 ubiquitin ligase. PROTAC Sirt2 Degrader-1 shows an IC50 of 0.25 μM for Sirt2, with no effect on Sirt1/Sirt3 (IC50s > 100 μM)[1]. |
Targets&IC50 | SIRT2:0.25 μM |
Molecular Weight | 852.94 |
Formula | C40H40N10O8S2 |
CAS No. | 2098487-75-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 100 mg/mL (117.24 mM)
You can also refer to dose conversion for different animals. More
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PROTAC Sirt2 Degrader-1 2098487-75-1 Chromatin/Epigenetic DNA Damage/DNA Repair Sirtuin PROTAC Sirt2 Degrader 1 PROTAC Sirt-2 Degrader-1 PROTAC Sirt2 Degrader1 inhibitor inhibit