Powder: -20°C for 3 years | In solvent: -80°C for 1 year
PF-4840154 is a potent, selective agonist of the rat and human TrpA1 channel and elicited TrpA1-mediated nocifensive behaviour in mouse, with EC50 of 97 nM and 23 nM for rTrpA1 and hTrpA1, respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
1 mg | In stock | $ 111.00 | |
2 mg | In stock | $ 160.00 | |
5 mg | In stock | $ 342.00 | |
10 mg | In stock | $ 497.00 | |
25 mg | In stock | $ 793.00 | |
50 mg | In stock | $ 1,130.00 | |
100 mg | In stock | $ 1,520.00 | |
1 mL * 10 mM (in DMSO) | In stock | $ 356.00 |
Description | PF-4840154 is a potent, selective agonist of the rat and human TrpA1 channel and elicited TrpA1-mediated nocifensive behaviour in mouse, with EC50 of 97 nM and 23 nM for rTrpA1 and hTrpA1, respectively. |
Targets&IC50 | hTRPA1:23 nM, rTRPA1:97 nM |
Molecular Weight | 466.62 |
Formula | C26H38N6O2 |
CAS No. | 1332708-14-1 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 4.66 mg/mL (10 mM)
You can also refer to dose conversion for different animals. More
bottom
Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc.
PF-4840154 1332708-14-1 Membrane transporter/Ion channel TRP/TRPV Channel licking nocifensive Inhibitor PF4840154 PF 4840154 non-electrophilic inhibit Transient receptor potential channels behavior TRP Channel inhibitor