1
Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T28269 | ORY-1001 free base | RG 6016 , ORY-1001 , ORY 1001 , ORY1001 , RG-6016 , RG6016 | |
ORY-1001 is a KDM1A inhibitor (IC50 <20nM) with high selectivity against related FAD dependent aminoxidases (MAO-A/B, IL4I1, KDM1B >100uM, SMOX 7uM). Treatment of THP-1 (MLL-AF9) cells with ORY-1001, results in a time/do... |