Powder: -20°C for 3 years | In solvent: -80°C for 1 year
NNC052090 is a GABA uptake inhibitor that displays moderate selectivity for BGT-1 transporters with Ki values are 1.4, 15, 19 and 41 μM for hBGT-1, hGAT-3, hGAT-1 and hGAT-2 respectively. NNC052090 also displays affinity at α1- and D2-receptors with IC50 values are 266 and 1632 nM respectively.
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 6-8 weeks | $ 1,520.00 | |
50 mg | 6-8 weeks | $ 1,980.00 | |
100 mg | 6-8 weeks | $ 2,500.00 |
Description | NNC052090 is a GABA uptake inhibitor that displays moderate selectivity for BGT-1 transporters with Ki values are 1.4, 15, 19 and 41 μM for hBGT-1, hGAT-3, hGAT-1 and hGAT-2 respectively. NNC052090 also displays affinity at α1- and D2-receptors with IC50 values are 266 and 1632 nM respectively. |
Synonyms | NNC-052090, NNC-05-2090, NNC05-2090, NNC 052090, NNC 05-2090 |
Molecular Weight | 414.54 |
Formula | C27H30N2O2 |
CAS No. | 184845-43-0 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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NNC052090 184845-43-0 NNC-052090 NNC-05-2090 NNC05-2090 NNC 052090 NNC 05-2090 inhibitor inhibit